Valsartan |
Diovan |
Image:Valsartan.png Valsartan Systematic (IUPAC) name 3-methyl-2- [pentanoyl-[ [4-[2-(2H-tetrazol-5-yl) phenyl] phenyl] methyl]amino] -butanoic acid Identifiers CAS number 137862-53-4 ATC code C09CA03 PubChem 60846 DrugBank APRD00133 Chemical data Formula C24H29N5O3 Mol. weight 435.519 g/mol Pharmacokinetic data Bioavailability ? Protein binding 95% Metabolism ? Half life 6 hours Excretion ? Therapeutic considerations Pregnancy cat. ...
Wikipedia - [full article]
Valsartan Clinical Trials
- A Study in Patients With Diabetes Mellitus Type II of the Effect on Albuminuria of 24 Week Treatment With Valsartan, Benazepril, and Valsartan+Benazepril
ClinicalTrials.gov Identifier: NCT00171119 - Active, not recruiting
Hypertension; Diabetic Nephropathy
- A Safety and Tolerability Study of the Combination of Aliskiren/Valsartan in Patients With High Blood Pressure, Followed by Long-Term Safety and Tolerability of Aliskiren, Valsartan and Hydrochlorothiazide.
ClinicalTrials.gov Identifier: NCT00386607 - Active, not recruiting
Hypertension
- Kanagawa Valsartan Trial (KVT): Effects of Valsartan on Renal and Cardiovascular Disease
ClinicalTrials.gov Identifier: NCT00190580 - Recruiting
Chronic Kidney Disease; Hypertension
- A Morbi-Mortality and Remodeling Study with Valsartan
ClinicalTrials.gov Identifier: NCT00133328 - Active, not recruiting
Hypertension; Ischemic Heart Disease; Congestive Heart Failure
- Valsartan in Cardiovascular Disease with Renal Dysfunction (The V-CARD) Study
ClinicalTrials.gov Identifier: NCT00140790 - Recruiting
Hypertension; Renal Dysfunction
- Safety and Efficacy of Valsartan Plus Hydrochlorothiazide and Amlodipine in Hypertensive Patients
ClinicalTrials.gov Identifier: NCT00426478 - Active, not recruiting
Hypertension
- Efficacy and Safety of Valsartan and the Combination of Valsartan and Simvastatin
ClinicalTrials.gov Identifier: NCT00385931 - Completed
Hypertension; Hypercholesterolemia; Dyslipidemia
- Valsartan/Hydrochlorothiazide Combination in Hypertensive Patients Not Controlled With Valsartan Alone
ClinicalTrials.gov Identifier: NCT00170989 - Completed
Hypertension
- Efficacy and Safety of Valsartan/Amlodipine Combination in Hypertensive Patients Not Controlled With Valsartan Alone
ClinicalTrials.gov Identifier: NCT00170963 - Completed
Hypertension
- Add-on Effects of Valsartan on Morbi- Mortality (KYOTO HEART Study)
ClinicalTrials.gov Identifier: NCT00149227 - Recruiting
Hypertension; Ischemic Heart Disease; Congestive Heart Failure; Stroke
- A Study to Describe Vascular and Renal Effects and Safety of Valsartan in Patients With High Blood Pressure
ClinicalTrials.gov Identifier: NCT00171353 - Active, not recruiting
Hypertension
- Safety and Efficacy of Valsartan Versus Atenolol and Hydrochlorothiazide Combination on Blood Flow in Hypertensive Patients
ClinicalTrials.gov Identifier: NCT00396656 - Active, not recruiting
Hypertension
- Comparison of Valsartan with Amlodipine in Hypertensive Patients with Glucose Intolerance
ClinicalTrials.gov Identifier: NCT00129233 - Recruiting
Hypertension; Type 2 Diabetes Mellitus; Impaired Glucose Tolerance
- Efficacy and Safety of Valsartan Versus Amlodipine in Postmenopausal Women With Hypertension
ClinicalTrials.gov Identifier: NCT00171054 - Active, not recruiting
Hypertension
- Efficacy and Safety of Valsartan/Hydrochlorothiazide Combination Therapy in Patients With Hypertension
ClinicalTrials.gov Identifier: NCT00277472 - Active, not recruiting
Hypertension
- Efficacy and Safety of Valsartan/Hydrochlorothiazide Combination Therapy in Patients With Hypertension
ClinicalTrials.gov Identifier: NCT00280540 - Active, not recruiting
Hypertension
- Efficacy and Safety of Valsartan, Hydrochlorothiazide and Amlodipine Combination Therapy in Hypertension
ClinicalTrials.gov Identifier: NCT00400777 - Active, not recruiting
Hypertension
- Efficacy and Safety of Valsartan and Amlodipine in Adults With Moderate, Inadequately Controlled Hypertension
ClinicalTrials.gov Identifier: NCT00523744 - Active, not recruiting
Hypertension
- Safety/Efficacy of Valsartan/Hydrochlorothiazide Combination Compared to Hydrochlorothiazide in Obese Hypertensive Adults
ClinicalTrials.gov Identifier: NCT00439738 - Active, not recruiting
Hypertension
- Safety and Efficacy of Enteric-Coated Mycophenolate Sodium (EC-MPS) Plus Valsartan in Patients With Kidney Transplants (MYTHOS
ClinicalTrials.gov Identifier: NCT00308425 - Active, not recruiting
De Novo Renal Transplantation
- A Clinical Study to Evaluate Safety & Efficacy of the Combination of Aliskiren, Valsartan & Hydrochlorothiazide in Diabetic Hypertensive Nonresponder Patients
ClinicalTrials.gov Identifier: NCT00219102 - Active, not recruiting
Hypertension; Diabetes
- Effects of Blood Pressure Reduction on High Sensitivity C-Reactive Protein (hsCRP)
ClinicalTrials.gov Identifier: NCT00154271 - Completed
Hypertension
- GISSI-AF - Use of Valsartan an Angiotensin II AT1-Receptor Blocker in the Prevention of Atrial Fibrillation Recurrence
ClinicalTrials.gov Identifier: NCT00376272 - Active, not recruiting
Atrial Fibrillation
- Long Term Study of Valsartan and Amlodipine in Patients With Essential Hypertension (Extension to Study CVAA489A1301)
ClinicalTrials.gov Identifier: NCT00446524 - Active, not recruiting
Hypertension
- Efficacy and Safety of Valsartan Versus Placebo on Exercise Tolerance in Patients With Heart Failure
ClinicalTrials.gov Identifier: NCT00171106 - Active, not recruiting
Diastolic Dysfunction, Symptomatic Heart Failure
- To Compare the Efficacy and Safety of TW vs Valsartan in the MN
ClinicalTrials.gov Identifier: NCT00518219 - Recruiting
Membranous Nephropathy
- To Compare the Efficacy and Safety of TW vs Valsartan in the DN
ClinicalTrials.gov Identifier: NCT00518362 - Recruiting
Diabetic Nephropathy
- Efficacy of Valsartan/Hydrochlorothiazide Versus Amlodipine and Hydrochlorothiazide in Patients Hypertension
ClinicalTrials.gov Identifier: NCT00425997 - Active, not recruiting
Hypertension
- Efficacy/Safety of Valsartan Plus Amlodipine and Amlodipine Alone in Patients With Hypertension
ClinicalTrials.gov Identifier: NCT00413049 - Active, not recruiting
Hypertension
- Efficacy/Safety of Valsartan Plus Amlodipine and Amlodipine Alone in Patients With Hypertension
ClinicalTrials.gov Identifier: NCT00413413 - Active, not recruiting
Hypertension
- Valsartan Optimal Therapy Against Elevated Home Blood Pressure Research(VOYAGER)Study
ClinicalTrials.gov Identifier: NCT00460213 - Recruiting
Hypertension
- A 10-12 Week Study to Evaluate the Safety and Efficacy of 320 mg Valsartan and 80 mg Simvastatin in Combination and as Monotherapies in Treating Hypertension and Hypercholesterolemia
ClinicalTrials.gov Identifier: NCT00171093 - Active, not recruiting
Hypertension; Hypercholesterolemia
- Open Label Extension Study to Evaluate the Long Term Use of Valsartan in 1-5 Year Old Hypertensive Children
ClinicalTrials.gov Identifier: NCT00457626 - Recruiting
Hypertension
- Safety and Efficacy of Valsartan/Amlodipine Compared to Amlodipine in Patients With Essential Hypertension
ClinicalTrials.gov Identifier: NCT00437645 - Active, not recruiting
Essential Hypertension
- Effectiveness of a Valsartan Based vs an Amlodipine Based Treatment Strategy in naïve Patients With Stage 1 or Stage 2 Hypertension or in Patients Uncontrolled on Current Monotherapy
ClinicalTrials.gov Identifier: NCT00351130 - Active, not recruiting
Hypertension
- A 16 Week Study to Evaluate the Effect on Insulin Sensitivity of Valsartan (320 mg) and Hydrochlorothiazide (25 mg) Combined and Alone, in Patients With Metabolic Syndrome
ClinicalTrials.gov Identifier: NCT00170937 - Active, not recruiting
Metabolic Syndrome; Hypertension; Pre-Hypertension
- Efficacy and Safety of Valsartan in Combination With Amlodipine Compared to Losartan Plus Hydrochlorothiazide in Patients With Hypertension and Left Ventricular Hypertrophy
ClinicalTrials.gov Identifier: NCT00446563 - Active, not recruiting
Hypertension; Hypertrophy, Left Ventricular
- A Study of the Antioxidant Probucol Combined With Valsartan in Patients With IgA Nephropathy
ClinicalTrials.gov Identifier: NCT00426348 - Recruiting
Glomerulonephritis, IGA
- Long Term Safety, Tolerability and Efficacy of Valsartan and Enalapril Combined and Alone in Children With Hypertension
ClinicalTrials.gov Identifier: NCT00446511 - Recruiting
Hypertension
- Pharmacokinetic Drug Interaction Study Following co-Administration of Valsartan, Hydrochlorothiazide and Amlodipine in Patients With Hypertension
ClinicalTrials.gov Identifier: NCT00548067 - Recruiting
Hypertension
- A Study of Valsartan Administered Once Daily Versus Twice Daily, in Patients With Stable, Chronic Heart Failure
ClinicalTrials.gov Identifier: NCT00294086 - Active, not recruiting
Chronic Heart Failure
- To Assess the Effects of Valsartan on Albuminuria/Proteinuria in Hypertensive Patients With Type 2 Diabetes Mellitus
ClinicalTrials.gov Identifier: NCT00550095 - Recruiting
Microalbuminuria; Proteinuria
- Efficacy of the New Closure Device in Improving Patient Compliance in Treatment of Hypertension With Valsartan+/-Hydrochlorothiazide (HCTZ) at 6 Months
ClinicalTrials.gov Identifier: NCT00487123 - Recruiting
Hypertension
- A Study to Compare Treating Hypertension With Valsartan 160 MG to Valsartan 320 Mg
ClinicalTrials.gov Identifier: NCT00241137 - Completed
Hypertension
- Telmisartan vs. valsartan missed dose
ClinicalTrials.gov Identifier: NCT00034840 - Completed
Hypertension
- To Compare the Blood Level of Marketed Japanese Valsartan Tablet Formulation vs Global Valsartan Tablet Formulation in Healthy Volunteers
ClinicalTrials.gov Identifier: NCT00415883 - Completed
Healthy
- Effect of Valsartan Compared to Enalapril on Sitting Systolic Blood Pressure in Children With High Blood Pressure
ClinicalTrials.gov Identifier: NCT00433836 - Recruiting
Hypertension
- Dose Response of Valsartan on Sitting Systolic Blood Pressure in 1-5 Year Old Children With High Blood Pressure
ClinicalTrials.gov Identifier: NCT00435162 - Recruiting
Hypertension
- Prevention of CHOP-Induced Chronic Cardiotoxicity
ClinicalTrials.gov Identifier: NCT00162955 - Recruiting
Non-Hodgkin''s Lymphoma
- Efficacy of Irbesartan/Hydrochlorothiazide Versus Valsartan/Hydrochlorothiazide in Mild to Moderate Hypertension
ClinicalTrials.gov Identifier: NCT00500604 - Recruiting
Hypertension
- Long-term Study of Starlix+Diovan to Delay Type II Diabetes Mellitus
ClinicalTrials.gov Identifier: NCT00097786 - Active, not recruiting
Diabetes Mellitus, Type 2
- Effect of Valsartan on Carotid Artery Disease
ClinicalTrials.gov Identifier: NCT00208767 - Recruiting
Carotid Artery Diseases; Atherosclerosis
- Efficacy and Safety of Valsartan and Amlodipine in Patients With Essential Hypertension
ClinicalTrials.gov Identifier: NCT00425373 - Recruiting
Essential Hypertension
- Efficacy and Safety of Aliskiren and Valsartan Versus Placebo in Patients Stabilized Following an Acute Coronary Syndrome
ClinicalTrials.gov Identifier: NCT00409578 - Recruiting
Post Acute Coronary Syndrome; Myocardial Ischemia
- The Effects of Systolic Blood Pressure Lowering on Diastolic Function Using Valsartan + Amlodipine in Patients With Hypertension and Diastolic Dysfunction
ClinicalTrials.gov Identifier: NCT00523549 - Recruiting
Hypertension; Diastolic Dysfunction
- Valsartan in Elderly Isolated Systolic Hypertension (VALISH) Study
ClinicalTrials.gov Identifier: NCT00151229 - Active, not recruiting
Elderly; Isolated Systolic Hypertension
- Effectiveness of Losartan 50 mg/HCTZ 12.5 mg Versus Valsartan 80 mg/HCTZ 12.5 mg Titrated as Needed in Patients With Hypertension Not Controlled on Monotherapy
ClinicalTrials.gov Identifier: NCT00546754 - Recruiting
Hypertension
- Effects of Continuous Positive Airway Pressure and Valsartan Treatments on Arterial Blood Pressure in OSAS Patients
ClinicalTrials.gov Identifier: NCT00409487 - Not yet recruiting
Hypertension,; Obstructive Sleep Apnea
- A Prospective, Randomised, Double-Blind, Double-Dummy, Forced-Titration, Multicentre, Parallel Group, One Year Treatment Trial to Investigate the Efficacy of Telmisartan 80 Mg Versus Valsartan 160 Mg in Hypertensive Type 2 Diabetic Patients with Overt Nep
ClinicalTrials.gov Identifier: NCT00153023 - Completed
Diabetic Nephropathies; Hypertension
- Antiproteinuric Effect of Valsartan and Lisinopril
ClinicalTrials.gov Identifier: NCT00171574 - Completed
Hypertension; Diabetic Nephropathy
- VALERIA: Valsartan in Combination With Lisinopril in Hypertensive Patients With Microalbuminuria
ClinicalTrials.gov Identifier: NCT00171067 - Completed
Hypertension
- Comparison of the Antihypertensive Efficacy of Valsartan and Enalapril After Missing One Dose
ClinicalTrials.gov Identifier: NCT00302705 - Completed
Hypertension
- A Study to Evaluate the Combination of Valsartan + Amlodipine in Hypertensive Patients
ClinicalTrials.gov Identifier: NCT00392262 - Completed
Hypertension
- Safety and Efficacy of Valsartan and Amlodipine Combined and Alone in Hypertensive Patients
ClinicalTrials.gov Identifier: NCT00409643 - Completed
Hypertension
- A Randomized, Double-Blind, Placebo-Controlled, Forced-Titration, Phase IV Study Comparing Telmisartan 80 Mg + Hydrochlorothiazide 25 Mg [Micardis HCT] Versus Valsartan 160 Mg + Hydrochlorothiazide 25 Mg [Diovan HCT] Taken Orally for Eight Weeks in Patien
ClinicalTrials.gov Identifier: NCT00168779 - Completed
Hypertension
- Comparison Of Morning And Evening Dosing Of Valsartan And Lisinopril In Patients With Diabetes
ClinicalTrials.gov Identifier: NCT00241124 - Completed
Hypertension
- VALORY Study of Valsartan/Hydrochlorizide for Patients Who do Not Respond Adequately to Olmesartan Medoxomil
ClinicalTrials.gov Identifier: NCT00171015 - Completed
Hypertension
- A Study to Evaluate the Combination of Valsartan and Amlodipine in Hypertensive Patients Not Controlled on Monotherapy
ClinicalTrials.gov Identifier: NCT00327145 - Completed
Hypertension
- VALENCE: Valsartan Versus Atenolol on Exercise Capacity in Hypertensive Overweight Postmenopausal Women
ClinicalTrials.gov Identifier: NCT00171132 - Completed
Hypertension
- Study to Compare the Effect of Valsartan vs Atenolol on Pro-Thrombotic State in Hypertensive Patients.
ClinicalTrials.gov Identifier: NCT00171756 - Completed
Hypertension
- VALIDATE Valsartan and Supportive Measures - Impact on Drug Adherence of Treated Hypertensive Patients
ClinicalTrials.gov Identifier: NCT00394823 - Completed
Hypertension
- Efficacy and Safety of Valsartan/Amlodipine Combination in Patients With Severe Hypertension
ClinicalTrials.gov Identifier: NCT00171535 - Completed
Hypertension
- Valsartan/Hydrochlorothiazide Combination vs Amlodipine in Patients With Hypertension, Diabetes, and Albuminuria.
ClinicalTrials.gov Identifier: NCT00171561 - Completed
Hypertension
- Safety and Efficacy of Valsartan and Amlodipine Combined and Alone in Patients With Hypertension.
ClinicalTrials.gov Identifier: NCT00409760 - Completed
Hypertension
- Efficacy and Safety of Valsartan/Amlodipine Combination in Hypertensive Patients Not Controlled With Amlodipine Alone
ClinicalTrials.gov Identifier: NCT00171002 - Completed
Hypertension
- One Year Study to Evaluate the Safety of the Combination of Valsartan and Amlodipine in Patients With Hypertension
ClinicalTrials.gov Identifier: NCT00409851 - Completed
Hypertension
- Bioavailability of Aliskiren and Valsartan Combined as a Single Tablet vs. the Same Medications Given Separately to Healthy Subjects.
ClinicalTrials.gov Identifier: NCT00416468 - Completed
Healthy
- Bioavailability of Aliskiren and Valsartan as a Single Tablet vs. the Same Doses of the Two Drugs Given Separately to Healthy Subjects.
ClinicalTrials.gov Identifier: NCT00416728 - Completed
Healthy
- A Study Comparing Valsartan With And Without Hydrochlorothiazide In Patients With Hypertension
ClinicalTrials.gov Identifier: NCT00241007 - Completed
Hypertension
- Valsartan/Hydrochlorothiazide Combination in the Treatment of Severe Hypertension
ClinicalTrials.gov Identifier: NCT00273299 - Completed
Hypertension
- Efficacy and Safety of Fluvastatin or Valsartan and Their Combination in Dyslipidemic Patients With Hypertension and Endothelial Dysfunction
ClinicalTrials.gov Identifier: NCT00171327 - Completed
Hypertension; Dyslipidemia
- A Study Of Valsartan Used To Treat Hypertension For Up To 13 Months In Hypertensive Children Ages 6 - 16 Years Of Age
ClinicalTrials.gov Identifier: NCT00171041 - Completed
Hypertension
- The Relative Effects of Olmesartan Medoxomil, Irbesartan and Valsartan on the Activity of the Blood Pressure Control System in Healthy Subjects
ClinicalTrials.gov Identifier: NCT00185055 - Completed
Healthy
- 8-Week Study to Evaluate Safety and Efficacy of Various Combinations of Valsartan, HCTZ, and Amlodipine in Patients With Moderate to Severe Hypertension
ClinicalTrials.gov Identifier: NCT00327587 - Completed
Hypertension
- Efficacy and Safety of the Combination of Valsartan Plus Amlodipine in Hypertensive Patients Not Adequately Responding to the Combination Therapy With Ramipril Plus Felodipine
ClinicalTrials.gov Identifier: NCT00367939 - Completed
Hypertension
- A Randomized, Double-Blind, Placebo Controlled Comparison of Telmisartan HCT and Valsartan HCT in HTN Stage I/II Patient
ClinicalTrials.gov Identifier: NCT00240448 - Completed
Hypertension
- Clinical Study to Evaluate Efficacy and Safety of Aliskiren (150mg & 300mg) Administered Alone and in Combo With Valsartan (160mg and 320mg) in Patients With High Blood Pressure
ClinicalTrials.gov Identifier: NCT00219180 - Completed
Hypertension
- A Study Of Valsartan Used To Treat Hypertension For Up To 56 Weeks In Children Ages 1 – 5 Years Who Have Hypertension
ClinicalTrials.gov Identifier: NCT00171028 - Completed
Hypertension
- VALID: Study to Compare the Reduction of Predialysis Systolic Blood Pressure With Valsartan Compared to Irbesartan in Patients With Mild to Moderate Hypertension on Long-Term Hemodialysis
ClinicalTrials.gov Identifier: NCT00171080 - Completed
Hypertension
- A Year Long Study to Evaluate the Safety of the Combination of Valsartan (320 mg) and Amlodipine (5 mg) in Patients With Hypertension
ClinicalTrials.gov Identifier: NCT00170976 - Completed
Hypertension
- The VALIDATE Study of Valsartan for Patients With Early Stage Heart Failure
ClinicalTrials.gov Identifier: NCT00241098 - Completed
Hypertension; Congestive Heart Failure
- Effect of Valsartan on Lipid Subfractions in Hypertensive Patients With Metabolic Syndrome
ClinicalTrials.gov Identifier: NCT00394745 - Completed
Hypertension; Metabolic Syndrome
- A Clinical Study to Evaluate the Safety and Efficacy of the Combination of Aliskiren and Valsartan in Hypertensive Non Responders Patients
ClinicalTrials.gov Identifier: NCT00219193 - Completed
Hypertension.
- Efficacy & Safety of Orally Administered Valsartan/Amlodipine Combo Therapy vs Amlodipine Monotherapy in Patients With Stage II Hypertension
ClinicalTrials.gov Identifier: NCT00350168 - Completed
Hypertension
- Efficacy & Safety of Orally Administered Valsartan/Amlodipine Combo Therapy vs Amlodipine Monotherapy in Black Patients With Stage II Hypertension
ClinicalTrials.gov Identifier: NCT00353912 - Completed
Hypertension
- Efficacy and Safety of Valsartan Plus Hydrochlorothiazide in Fixed Dose Combination in Hypertensive Patients Not Controlled by the Free Combination of an Angiotensin Receptor Blocker Plus Hydrochlorothiazide
ClinicalTrials.gov Identifier: NCT00360178 - Completed
Hypertension
- Diva - The Effects Of 12 Weeks Of Treatment With High Dose Valsartan (320 Mg) To Amlodipine On Endothelial Function In Hypertensive Subjects With The Metabolic Syndrome
ClinicalTrials.gov Identifier: NCT00241150 - Completed
Hypertension; Metabolic Syndrome
- Comparative Study of Valsartan and Amlodipine Versus Amlodipine Alone in Hypertension
ClinicalTrials.gov Identifier: NCT00333489 - Completed
Hypertension
- Clinical Trial To Evaluate The Effect Of Valsartan On Insulin Sensitivity In Subjects With Impaired Glucose Tolerance
ClinicalTrials.gov Identifier: NCT00241072 - Completed
Hypertension; Impaired Glucose Tolerance
- A Study to Evaluate the Efficacy of Valsartan/Simvastatin Combinations in Patients With Both Essential Hypertension and Hypercholesterolemia
ClinicalTrials.gov Identifier: NCT00254475 - Completed
Essential Hypertension; Hypercholesterolemia

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